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6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists

Wei Sun1, Hyo-Shin Kim2, Sunho Lee2

  • 1Shenyang Pharmaceutical University, Shenyang 110016, China; Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|January 19, 2015
PubMed

Keywords:
AnalgesicMolecular modelingTRPV1 antagonistVanilloid receptor 1

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