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Discovery and structure-activity relationship studies of N6-benzoyladenine derivatives as novel BRD4 inhibitors

Tomomi Noguchi-Yachide1, Taki Sakai1, Yuichi Hashimoto1

  • 1Institute of Molecular and Cellular, Biosciences, The University of Tokyo, 1-1-1 Yayoi, Bunkyo-ku, Tokyo 113-0032, Japan.

Bioorganic & Medicinal Chemistry
|February 14, 2015
PubMed

Keywords:
BRD4BenzoyladenineBromodomainStructure–activity relationship

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