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PDK1 disruptors and modulators: a patent review

Muhammad Jahangir Hossen1, Seung Cheol Kim, Sungjae Yang

  • 1Sungkyunkwan University, Department of Genetic Engineering , 300 Chuncheon-Dong, Suwon 440-746 , Korea +82 31 290 7868 ; +82 31 290 7870 ; jaecho@skku.edu.

Expert Opinion on Therapeutic Patents
|February 17, 2015
PubMed
Summary

3-Phosphoinositide-dependent kinase 1 (PDK1) is a key regulator in cancer. Research focuses on developing small molecule PDK1 inhibitors and modulators, with over 50 patents published since 1998.

Keywords:
3-phosphoinositide-dependent kinase 13-phosphoinositide-dependent kinase 1 inhibitors3-phosphoinositide-dependent kinase 1 modulators

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