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Atracurium and vecuronium interaction with gentamicin and tobramycin

J Y Dupuis1, R Martin, J P Tétrault

  • 1Department of Anaesthesia, University of Sherbrooke, P. Que.

Insights

Aminoglycoside antibiotics like tobramycin and gentamicin prolong neuromuscular blockade from vecuronium but not atracurium. Atracurium may be a safer choice for patients on these antibiotics when prolonged block is not desired.

Area of Science:

  • Pharmacology
  • Anesthesiology
  • Critical Care Medicine

Background:

  • Aminoglycosides are commonly used antibiotics.
  • Neuromuscular blocking agents are used in anesthesia and critical care.
  • Potential drug interactions between these classes require investigation.

Purpose of the Study:

  • To investigate the interaction between aminoglycosides (tobramycin, gentamicin) and neuromuscular blocking agents (atracurium, vecuronium).
  • To determine if therapeutic aminoglycoside levels affect the onset, duration, and recovery of neuromuscular blockade.

Main Methods:

  • Prospective study in 44 patients.
  • 22 patients with therapeutic aminoglycoside levels vs. 22 controls.
  • Measured onset time, clinical duration, and recovery time of neuromuscular blockade after atracurium or vecuronium administration.

Main Results:

  • No significant difference in onset time for either drug.
  • Vecuronium's clinical duration and recovery time were significantly prolonged in patients receiving aminoglycosides (P<0.01 and P<0.0005, respectively).
  • Atracurium's neuromuscular block was not significantly affected by aminoglycoside therapy.

Conclusions:

  • Aminoglycosides prolong vecuronium-induced neuromuscular blockade.
  • Atracurium's neuromuscular blockade is not significantly influenced by aminoglycosides.
  • Atracurium may offer an advantage over vecuronium in patients receiving aminoglycosides when a prolonged block is undesirable.

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