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Pharmacokinetic, pharmacodynamic and metabolic characterization of a brain retentive microtubule (MT)-stabilizing

Anne-Sophie Cornec1, Michael J James2, Jane Kovalevich2

  • 1Department of Chemistry, School of Arts and Sciences, University of Pennsylvania, 231 South 34th St., Philadelphia, PA 19104-6323, United States.

Bioorganic & Medicinal Chemistry Letters
|March 31, 2015
PubMed

Keywords:
CNS drug discoveryMicrotubule stabilizationPharmacodynamicPharmacokineticTriazolopyrimidine

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