[11C]PBR28 PET imaging is sensitive to neuroinflammation in the aged rat

Matthew D Walker1, Katherine Dinelle2, Rick Kornelsen2

  • 1Department of Physics and Astronomy, University of British Columbia, Vancouver, British Columbia, Canada.

Insights

Brain imaging with [(11)C]PBR28 shows increased microglial activation in aging rats. This neuroinflammation marker rises with age, regardless of Parkinson's disease risk genes, suggesting aging itself drives these changes.

Area of Science:

  • Neuroscience
  • Radiochemistry
  • Gerontology

Background:

  • Aging is associated with increased neuroinflammation, a key factor in neurodegenerative diseases.
  • Microglial activation is a primary indicator of neuroinflammation.
  • Positron Emission Tomography (PET) imaging offers a non-invasive method to study brain changes in vivo.

Purpose of the Study:

  • To investigate age-related changes in neuroinflammation using [(11)C]PBR28 PET imaging in rats.
  • To assess the impact of the LRRK2 p.G2019S mutation, a risk factor for Parkinson's disease, on age-related neuroinflammation.
  • To correlate in vivo PET findings with in vitro autoradiography data.

Main Methods:

  • Utilized [(11)C]PBR28 microPET imaging in normal and LRRK2 p.G2019S transgenic rats across different ages.
  • Acquired 70 PET scans and performed arterial blood sampling for tracer kinetic modeling to estimate total volume of distribution (VT).
  • Conducted in vitro autoradiography to validate PET findings and measured plasma free fraction (fp).

Main Results:

  • [(11)C]PBR28 uptake in the brain significantly increased with age in both normal and transgenic rats.
  • Standard Uptake Value (SUV) increased by 56% and VT by 91% over 12 months of aging (4 to 16 months).
  • In vitro binding showed a 19% increase with aging (4 to 20 months), correlating with PET data.

Conclusions:

  • Brain uptake of [(11)C]PBR28, a marker of microglial activation, increases with age in rats.
  • Aging, rather than the LRRK2 p.G2019S mutation, appears to be the primary driver of increased neuroinflammation in this model.
  • These findings highlight the utility of [(11)C]PBR28 PET imaging for studying age-related neuroinflammation.

Related Concept Videos