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Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions
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Efficient regioselective ring opening of activated aziridine-2-carboxylates with [(18)f]fluoride

Christina Schjoeth-Eskesen1, Paul Robert Hansen2, Andreas Kjaer3

  • 1Department of Clinical Physiology, Nuclear Medicine & PET, Copenhagen University Hospital Rigshospitalet Blegdamsvej 9, 2100 Copenhagen Ø (Denmark) ; Department of Clinical Physiology, Nuclear Medicine & PET, Copenhagen University Hospital Rigshospitalet Blegdamsvej 9, 2100 Copenhagen Ø (Denmark).

Chemistryopen
|April 11, 2015
PubMed

Keywords:
aziridinesfluorine-18radiochemistryregioselectivityring opening

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