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Updated: Apr 15, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Evolution and synthesis of novel orally bioavailable inhibitors of PDE10A

Douglas F Burdi1, John E Campbell1, Jun Wang1

  • 1Sunovion Pharmaceuticals Inc., 84 Waterford Drive, Marlborough, MA 01752, United States.

Bioorganic & Medicinal Chemistry Letters
|April 13, 2015
PubMed

Keywords:
PCP-induced hyperlocomotionPDE10APDE10A inhibitorPhosphodiesterase inhibitorSchizophrenia

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