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ABL kinase inhibitory and antiproliferative activity of novel picolinamide based benzothiazoles

Ashraf Kareem El-Damasy1, Nam-Chul Cho2, Soon Bang Kang3

  • 1Center for Neuro-Medicine, Brain Science Institute, Korea Institute of Science and Technology (KIST), Hwarangro 14-gil 5, Seongbuk-gu, Seoul 136-791, Republic of Korea; Department of Biological Chemistry, Korea University of Science and Technology (UST), Gajungro 217, Youseong-gu, Daejeon 305-350, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|April 18, 2015
PubMed

Keywords:
ABL kinaseAntiproliferativeBenzothiazoleChronic myelogenous leukemiaPicolinamideT315I mutant

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