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Exploring the isoform selectivity of TGX-221 related pyrido[1,2-a]pyrimidinone-based Class IA PI 3-kinase inhibitors:

Andrew J Marshall1, Claire L Lill2, Mindy Chao1

  • 1Auckland Cancer Society Research Centre, Faculty of Medical and Health Sciences, The University of Auckland, Private Bag 92019, Auckland 1142, New Zealand.

Bioorganic & Medicinal Chemistry
|April 20, 2015
PubMed

Keywords:
Comparative modellingDockingPI3KPhosphatidylinositol 3-kinaseTGX-221p110β

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