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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Synthesis and molecular docking of 1,2,3-triazole-based sulfonamides as aromatase inhibitors

Ratchanok Pingaew1, Veda Prachayasittikul2, Prasit Mandi3

  • 1Department of Chemistry, Faculty of Science, Srinakharinwirot University, Bangkok 10110, Thailand.

Bioorganic & Medicinal Chemistry
|May 3, 2015
PubMed

Keywords:
Anti-aromatase activityMolecular dockingStructure–activity relationshipsSulfonamideTetrahydroisoquinolineTriazole

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