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α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists

Phuong-Thao Tran1, Ho Shin Kim1, Jihyae Ann1

  • 1Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|May 5, 2015
PubMed

Keywords:
AnalgesicCapsaicinMolecular modelingTRPV1 antagonist

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