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Updated: Apr 12, 2026

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications
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Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications

Published on: January 27, 2014

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Gα(i/o)-coupled receptor-mediated sensitization of adenylyl cyclase: 40 years later

Tarsis F Brust1, Jason M Conley1, Val J Watts1

  • 1Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, 575 Stadium Mall Drive, West Lafayette, IN 47907, USA.

European Journal of Pharmacology
|May 19, 2015
PubMed

Keywords:
Adenylyl cyclaseG protein subunitG protein-coupled receptorHeterologous sensitizationProtein kinaseSuperactivation

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