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Discovery of a Potent Class of PI3Kα Inhibitors with Unique Binding Mode via Encoded Library Technology (ELT)

Hongfang Yang1, Patricia F Medeiros1, Kaushik Raha2

  • 1MDR (Molecular Discovery Research) Boston, Platform Technology and Science, GlaxoSmithKline , 830 Winter Street, Waltham, Massachusetts 02451, United States.

ACS Medicinal Chemistry Letters
|May 26, 2015
PubMed

Keywords:
ELTEncoded Library technologyPI3K p110α (H1047R)PI3Kαp110α

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