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Updated: Apr 11, 2026

Assays for Validating Histone Acetyltransferase Inhibitors
Published on: August 6, 2020
Alokta Chakrabarti1, Ina Oehme2, Olaf Witt3
1Institute of Pharmaceutical Sciences, Albert-Ludwigs-Universität Freiburg, Freiburg, Germany.
Histone deacetylase 8 (HDAC8) is a promising drug target for cancer, intellectual disability, and infections. Developing selective HDAC8 inhibitors is key to minimizing side effects compared to broad-acting drugs.
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