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A Michael Equilibration Model To Control Site Selectivity in the Condensation toward Aminopyrazoles

Daniel R Fandrick1, Sanjit Sanyal1, Joseph Kaloko1

  • 1†Chemical Development, Boehringer Ingelheim Pharmaceuticals, Inc., 900 Ridgebury Road, P.O. Box 368, Ridgefield, Connecticut 06877-0368, United States.

Organic Letters
|June 2, 2015
PubMed

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