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Discovery of novel pyrazole-containing benzamides as potent RORγ inverse agonists

Tao Wang1, Daliya Banerjee2, Tonika Bohnert1

  • 1Chemistry and Molecular Therapeutics, Biogen, 12 Cambridge Center, Cambridge, MA 02142, USA.

Bioorganic & Medicinal Chemistry Letters
|June 7, 2015
PubMed

Keywords:
Autoimmune diseaseIL-17InflammationRORγ inverse agonistTh17 cell

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