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CETSA: a target engagement assay with potential to transform drug discovery

Annika Jenmalm Jensen1, Daniel Martinez Molina2, Thomas Lundbäck1

  • 1Division of Translational Medicine & Chemical Biology, Department of Medical Biochemistry & Biophysics, Karolinska Institutet, Tomtebodavägen 23A, 171 65 Solna, Sweden.

Future Medicinal Chemistry
|June 12, 2015
PubMed
Abstract

No abstract available in PubMed .

Keywords:
CETSAR&D efficiencycellular thermal shift assayphenotypic-based drug-discoverytarget engagementtarget-based drug-discovery

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