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Updated: Apr 10, 2026

Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs
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Structure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors

Xu Ran1, Yujun Zhao1, Liu Liu1

  • 1†Departments of Medicinal Chemistry, ‡Internal Medicine, §Pharmacology, and ∥Biological Chemistry, ⊥Life Sciences Institute, and #Comprehensive Cancer Center, University of Michigan, Ann Arbor, Michigan 48109, United States.

Journal of Medicinal Chemistry
|June 17, 2015
PubMed

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