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Updated: Apr 6, 2026

Detecting the Ligand-binding Domain Dimerization Activity of Estrogen Receptor Alpha Using the Mammalian Two-Hybrid Assay
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Structural development of stabilized helical peptides as inhibitors of estrogen receptor (ER)-mediated transcription

Yosuke Demizu1, Takashi Misawa1, Takaya Nagakubo2

  • 1Division of Organic Chemistry, National Institute of Health Sciences, 1-18-1, Kamiyoga, Setagaya, Tokyo 158-8501, Japan.

Bioorganic & Medicinal Chemistry
|July 18, 2015
PubMed

Keywords:
Estrogen receptorHelical peptideProtein–protein interactionTranscriptional inhibitor

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