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Updated: Apr 6, 2026

Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors
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Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors

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Design and synthesis of new non nucleoside inhibitors of DNMT3A

Alexandre Erdmann1, Yoann Menon1, Christina Gros1

  • 1Unité de Service et de Recherche CNRS-Pierre Fabre n°3388, ETaC, CRDPF, 3 Avenue Hubert Curien, 31100 Toulouse, France.

Bioorganic & Medicinal Chemistry
|July 30, 2015
PubMed

Keywords:
DNA methylationDNMT3AMichael acceptorReactive inhibitor

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