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Discovery of N-(4-aryl-5-aryloxy-thiazol-2-yl)-amides as potent RORγt inverse agonists

Yonghui Wang1, Ting Yang2, Qian Liu2

  • 1School of Pharmacy, Fudan University, 826 Zhangheng Road, Pudong, Shanghai 201203, China.

Bioorganic & Medicinal Chemistry
|August 17, 2015
PubMed

Keywords:
Crystal structureRORγt inverse agonistsTh17 cell differentiationThiazole ether amides

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