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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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Synthesis and evaluation of arylpiperazine-reverse amides as biased dopamine D3 receptor ligands

Yongkai Cao1, Suresh Paudel1, Xiaowei Zhang1

  • 1College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 500-757, Republic of Korea.

Bioorganic & Medicinal Chemistry
|August 18, 2015
PubMed

Keywords:
Dopamine D3 receptorMolecular modelingReverse amideSelectivityStructure–activity relationships

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