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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Structures of G protein-coupled receptors reveal new opportunities for drug discovery

Robert M Cooke1, Alastair J H Brown1, Fiona H Marshall1

  • 1Heptares Therapeutics, Biopark, Broadwater Road, Welwyn Garden City, Hertfordshire AL7 3AX, UK.

Drug Discovery Today
|August 26, 2015
PubMed

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