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Assessment of Morphine-induced Hyperalgesia and Analgesic Tolerance in Mice Using Thermal and Mechanical Nociceptive Modalities
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Design, synthesis, and evaluation of new endomorphin analogs with enhanced central antinociception after peripheral

Xin Liu1, Long Zhao1, Yuan Wang1

  • 1Department of pharmacology, Key Laboratory of Preclinical Study for New Drugs of Gansu Province, Institute of Biochemistry and Molecular Biology, School of Basic Medical Sciences, School of Life Science, Lanzhou University, Lanzhou 730000, PR China.

Bioorganic & Medicinal Chemistry Letters
|September 26, 2015
PubMed

Keywords:
AnalgesiaBlood–brain barrierEndomorphinUnnatural amino acid

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