Chiral Inhibition of Rivaroxaban Derivatives Towards UDP-Glucuronosyltransferase (UGT) Isoforms

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Screening Traditional Chinese Medicine Compounds for Inhibiting UCHL3 Activity Based on Molecular Docking and Deubiquitinating Enzyme Probe Technology
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Screening Traditional Chinese Medicine Compounds for Inhibiting UCHL3 Activity Based on Molecular Docking and Deubiquitinating Enzyme Probe Technology

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Zhuhua Yao1, Yong-Zhe Liu2, Ai-Lun Ma3

  • 1Department of Cardiology, Tianjin Union Medicine Centre, 300121, Tianjin, People's Republic of China.

Chirality
|October 2, 2015
PubMed

Keywords:
UDP-glucuronosyltransferases (UGTs)chiralitydrug-drug interactionrivaroxaban

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