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Nitrofuranyl Methyl Piperazines as New Anti-TB Agents: Identification, Validation, Medicinal Chemistry, and PK

Kushalava Reddy Yempalla1, Gurunadham Munagala1, Samsher Singh1

  • 1Medicinal Chemistry Division, Clinical Microbiology Division, PK-PD and Toxicology Division, Pre-formulation Laboratory, Academy of Scientific and Innovative Research, CSIR-Indian Institute of Integrative Medicine , Canal Road, Jammu 180 001, India.

ACS Medicinal Chemistry Letters
|October 22, 2015
PubMed

Keywords:
6-nitro-2,3-dihydroimidazooxazoleMTB H37RvMycobacterium tuberculosismultidrug resistant-TBstructure−activity relationship

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