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Updated: Mar 30, 2026

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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Competitive Binding Assay for the G-Protein-Coupled Receptor 30 (GPR30) or G-Protein-Coupled Estrogen Receptor (GPER)

Thomas Thekkumkara1, Russell Snyder2, Vardan T Karamyan3

  • 1Department of Biomedical Sciences, Texas Tech University Health Sciences Center, 1300 Coulter Drive, Amarillo, TX, 79106, USA. thomas.thekkumkara@ttuhsc.edu.

Methods in Molecular Biology (Clifton, N.J.)
|November 21, 2015
PubMed

Keywords:
2-MethoxyestradiolCompetitive bind ingEndoplasmic reticulum membraneG-protein-coupled estrogen receptorG-protein-coupled receptor 30GPERGPR30Radioligand bind ing

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