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Synthesis of (3S,4S)-4-aminopyrrolidine-3-ol derivatives and biological evaluation for their BACE1 inhibitory

Quang De Tran1, Sukumar Bepary2, Ge Hyeong Lee2

  • 1Department of Medicinal and Pharmaceutical Chemistry, Korea University of Science and Technology, 217 Gajeong-ro, Yuseong-gu, Daejeon 305-333, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|November 27, 2015
PubMed

Keywords:
Alzheimer’s diseaseBACE1 inhibitorsPyrrolidine derivatives

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