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Identification of azabenzimidazoles as potent JAK1 selective inhibitors

Melissa M Vasbinder1, Marat Alimzhanov1, Martin Augustin2

  • 1AstraZeneca R&D Boston, Oncology IMED, 35 Gatehouse Drive, Waltham, MA 02451, United States.

Bioorganic & Medicinal Chemistry Letters
|November 29, 2015
PubMed

Keywords:
AzabenzimidazolesJAK selectivityJAK1JAK1 inhibitors

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