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Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions

Published on: November 30, 2022

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A novel protocol for the one-pot borylation/Suzuki reaction provides easy access to hinge-binding groups for kinase

A Hooper1, A Zambon, C J Springer

  • 1The Institute of Cancer Research, Cancer Research UK Cancer Therapeutics Unit, Division of Cancer Therapeutics, 15 Cotswold Road, Sutton, Surrey SM2 5NG, UK. Caroline.Springer@icr.ac.uk.

Organic & Biomolecular Chemistry
|December 2, 2015
PubMed

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