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Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Development of a novel sulfonate ester-based prodrug strategy

Kengo Hanaya1, Shohei Yoshioka1, Shinya Ariyasu2

  • 1Faculty of Pharmacy, Keio University, 1-5-30 Shibakoen, Minato-ku, Tokyo 105-8512, Japan.

Bioorganic & Medicinal Chemistry Letters
|December 9, 2015
PubMed

Keywords:
ProdrugProteaseSuicide substrateSulfonateSultam

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