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Synthesis, structure-activity relationship and biological evaluation of novel arylpiperzines as α1A/1D-AR

Fang Xu1, Hong Chen2, Jingyi Xu3

  • 1Institute of Tumor Pharmacology, College of Pharmacy, Jinan University, 601 West Huangpu Blvd, Guangzhou 510632, People's Republic of China.

Bioorganic & Medicinal Chemistry
|December 9, 2015
PubMed

Keywords:
Antagonic activityArylpiperazine derivativesHomology modelingStructure–activity relationshipSubtype selectivityα(1)-ARs

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