Farnesoid X Receptor Protects against Kidney Injury in Uninephrectomized Obese Mice
Zhibo Gai1, Ting Gui2, Christian Hiller1
1From the Department of Clinical Pharmacology and Toxicology, University Hospital Zurich, University of Zurich, CH-8091 Zurich, Switzerland and.
Abstract:
Activation of the farnesoid X receptor (FXR) has indicated a therapeutic potential for this nuclear bile acid receptor in the prevention of diabetic nephropathy and obesity-induced renal damage. Here, we investigated the protective role of FXR against kidney damage induced by obesity in mice that had undergone uninephrectomy, a model resembling the clinical situation of kidney donation by obese individuals. Mice fed a high-fat diet developed the core features of metabolic syndrome, with subsequent renal lipid accumulation and renal injury, including glomerulosclerosis, interstitial fibrosis, and albuminuria. The effects were accentuated by uninephrectomy. In human renal biopsies, staining of 4-hydroxynonenal (4-HNE), glucose-regulated protein 78 (Grp78), and C/EBP-homologous protein, markers of endoplasmic reticulum stress, was more prominent in the proximal tubules of 15 obese patients compared with 16 non-obese patients. In mice treated with the FXR agonist obeticholic acid, renal injury, renal lipid accumulation, apoptosis, and changes in lipid peroxidation were attenuated. Moreover, disturbed mitochondrial function was ameliorated and the mitochondrial respiratory chain recovered following obeticholic acid treatment. Culturing renal proximal tubular cells with free fatty acid and FXR agonists showed that FXR activation protected cells from free fatty acid-induced oxidative stress and endoplasmic reticulum stress, as denoted by a reduction in the level of reactive oxygen species staining and Grp78 immunostaining, respectively. Several genes involved in glutathione metabolism were induced by FXR activation in the remnant kidney, which was consistent with a decreased glutathione disulfide/glutathione ratio. In summary, FXR activation maintains endogenous glutathione homeostasis and protects the kidney in uninephrectomized mice from obesity-induced injury.
Insights
Activation of the farnesoid X receptor (FXR) protects kidneys from obesity-induced damage. FXR activation maintains glutathione homeostasis and reduces endoplasmic reticulum stress, offering a potential therapeutic strategy for kidney disease.
Area of Science:
- Nephrology
- Metabolic Syndrome
- Molecular Biology
Background:
- Obesity contributes to kidney damage, particularly in individuals with reduced renal mass.
- Obesity-induced kidney injury involves metabolic syndrome features, renal lipid accumulation, and endoplasmic reticulum stress.
- FXR (farnesoid X receptor) is a nuclear bile acid receptor with potential therapeutic applications.
Purpose of the Study:
- To investigate the protective role of FXR against obesity-induced kidney damage in a mouse model.
- To explore the effects of FXR activation on renal lipid accumulation, endoplasmic reticulum stress, and mitochondrial function.
- To assess the impact of FXR on glutathione homeostasis in the context of kidney injury.
Main Methods:
- Utilized a uninephrectomized mouse model fed a high-fat diet to induce obesity and kidney injury.
- Administered the FXR agonist obeticholic acid to treated mice.
- Analyzed human renal biopsies for markers of endoplasmic reticulum stress.
- Performed in vitro studies using renal proximal tubular cells exposed to free fatty acids and FXR agonists.
Main Results:
- High-fat diet and uninephrectomy exacerbated renal injury, lipid accumulation, and endoplasmic reticulum stress.
- Obeticholic acid treatment attenuated renal injury, lipid accumulation, apoptosis, and oxidative stress.
- FXR activation improved mitochondrial function and recovered the mitochondrial respiratory chain.
- FXR activation induced glutathione metabolism genes and maintained glutathione homeostasis.
Conclusions:
- FXR activation demonstrates a protective effect against obesity-induced kidney injury in a mouse model.
- FXR plays a crucial role in mitigating endoplasmic reticulum stress, oxidative stress, and lipid accumulation in the kidney.
- FXR activation supports endogenous glutathione homeostasis, contributing to renal protection.
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