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Testing Targeted Therapies in Cancer using Structural DNA Alteration Analysis and Patient-Derived Xenografts
Published on: July 25, 2020
Whole-exome tumor sequencing study in biliary cancer patients with a response to MEK inhibitors
Daniel H Ahn1, Hatice Gulcin Ozer2, Baris Hancioglu2
1Department of Internal Medicine, Divison of Medical Oncology, Ohio State University Comprehensive Cancer Center, Columbus, OH, USA.
Abstract:
We previously conducted a phase-II study with selumetinib (AZD6244), a small molecule inhibitor of MEK1/2, in advanced biliary tract cancers (BTC), where the primary endpoint was response rate. Several patients experienced objective response. These findings were confirmed with MEK162 in a similar patient population. To assess for tumor-specific genetic variants that mediate sensitivity to MEK inhibition in BTC, we performed whole-exome sequencing in patients with an objective response to selumetinib. Normal and tumor DNA from FFPE tissue from two patients who experienced an objective response underwent whole-exome sequencing. Raw sequence reads were processed with GATK workflow and tumor specific variants were identified using MuTect and VarScan2. Ensemble Variant Effect Predictor was used to determine functional consequences of these variants. Copy number changes and potential gene fusion events were also screened. Findings were compared to assess for any commonality between the two tumor samples, and whether the identified variants were intrinsic to the MAPK pathway. 1169 and 628 tumor-specific variants were identified in the two samples. Further analysis demonstrated 60 and 53 functional and novel variants, respectively. Of the identified tumor-specific variants, fusion events or copy number changes, no commonality was seen. Several variants in genes associated with ERK signaling were present in each tumor sample. Although there were no common tumor-specific variants in the two patients who exhibited an objective response to selumetinib, several genes associated with ERK signaling were identified. Confirmatory studies investigating the role of the identified genes and other potential tumor independent factors need further investigation.
Insights
Investigating MEK inhibitors in biliary tract cancers (BTC) revealed ERK signaling pathway variants. While no common tumor-specific mutations were found in responders, further studies are needed to confirm these genetic factors.
Area of Science:
- Oncology
- Genetics
- Pharmacology
Background:
- Biliary tract cancers (BTC) are aggressive malignancies with limited treatment options.
- Selumetinib, a MEK1/2 inhibitor, has shown activity in advanced BTC.
- Identifying genetic drivers of response to MEK inhibition is crucial for personalized therapy.
Purpose of the Study:
- To identify tumor-specific genetic variants associated with response to selumetinib in BTC.
- To investigate the role of the MAPK/ERK signaling pathway in BTC sensitivity to MEK inhibition.
Main Methods:
- Whole-exome sequencing of tumor and normal DNA from two BTC patients who responded to selumetinib.
- Bioinformatic analysis using GATK, MuTect, and VarScan2 to identify somatic variants.
- Functional consequence prediction using Ensemble Variant Effect Predictor and screening for copy number changes and gene fusions.
Main Results:
- 1169 and 628 tumor-specific variants were identified in the two samples, with 60 and 53 functional/novel variants respectively.
- No common tumor-specific variants, copy number changes, or gene fusions were found between the two responsive patients.
- Several variants in genes associated with ERK signaling were identified in both tumor samples.
Conclusions:
- While no shared genetic alterations were identified, the presence of ERK signaling pathway variants suggests its involvement in selumetinib response in BTC.
- Further research is warranted to elucidate the role of these identified genes and other potential factors in mediating sensitivity to MEK inhibition in BTC.
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