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Bromodomains: Structure, function and pharmacology of inhibition

Elena Ferri1, Carlo Petosa2, Charles E McKenna1

  • 1Department of Chemistry, Dana and David Dornsife College of Letters, Arts and Sciences, University of Southern California, University Park Campus, Los Angeles, CA 90089, United States.

Biochemical Pharmacology
|December 29, 2015
PubMed

Keywords:
Acetylated histonesBET proteinsBromodomainsDrug discoveryEpigenetic drugs

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