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Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay

Takayoshi Kinoshita1, Hajime Sugiyama2, Yurika Mori1

  • 1Graduate School of Science, Osaka Prefecture University, 1-1 Gakuen-cho, Naka-ku, Sakai, Osaka 599-8531, Japan.

Bioorganic & Medicinal Chemistry Letters
|January 7, 2016
PubMed

Keywords:
Allosteric inhibitorCompetitive binding assayCrystal structureERK2In silico screening

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