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Updated: Mar 27, 2026

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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Metal-Free Synthesis of Fluorinated Indoles Enabled by Oxidative Dearomatization

Edon Vitaku1, David T Smith1, Jon T Njardarson2

  • 1Department of Chemistry and Biochemistry, University of Arizona, 1306 E. University Blvd., Tucson, AZ, 85721, USA.

Angewandte Chemie (International Ed. in English)
|January 11, 2016
PubMed

Keywords:
dearomatizationfluorineindolesnitrogen heterocyclesynthetic methods

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