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Updated: Mar 27, 2026

Bio-layer Interferometry for Measuring Kinetics of Protein-protein Interactions and Allosteric Ligand Effects
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Molecular insights to the bioactive form of BV02, a reference inhibitor of 14-3-3σ protein-protein interactions

Daniela Valensin1, Ylenia Cau1, Pierpaolo Calandro1

  • 1Dipartimento di Biotecnologie, Chimica e Farmacia, Università degli studi di Siena, via A. Moro snc, Via Aldo Moro 2, 53100 Siena, Italy.

Bioorganic & Medicinal Chemistry Letters
|January 18, 2016
PubMed

Keywords:
14-3-3Bioactive formChemical instabilityChemical transformationDrug discoveryLead compoundNMR

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