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Updated: Mar 26, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Discovery of a Potent and Orally Efficacious TGR5 Receptor Agonist

Sameer Agarwal1, Amit Patil1, Umesh Aware1

  • 1Zydus Research Centre, Cadila Healthcare Ltd. , Sarkhej-Bavla N.H. No. 8 A, Moraiya, Ahmedabad 382 210, India.

ACS Medicinal Chemistry Letters
|January 29, 2016
PubMed

Keywords:
GLP1 secretionGPBAR1GPR 131TGR5TGR5 agonistdiabetes

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