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Updated: Mar 26, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Recent updates on GPCR biased agonism

André S Pupo1, Diego A Duarte2, Vanessa Lima3

  • 1Department of Pharmacology, Instituto de Biociências, UNESP, Botucatu, SP, Brazil.

Pharmacological Research
|February 3, 2016
PubMed

Keywords:
7TMRFunctional selectivityGPCR

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