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2-Oxo-1,2-dihydropyridinyl-3-yl amide-based GPa inhibitors: Design, synthesis and structure-activity relationship

Wendy A Loughlin1, Ian D Jenkins2, N David Karis2

  • 1School of Natural Sciences, Griffith University, Brisbane, QLD, 4111, Australia.

European Journal of Medicinal Chemistry
|February 8, 2016
PubMed

Keywords:
Glycogen phosphorylase inhibitorsPeptide mimeticPyridone amidesStructure activity relationshipType 2 diabetes

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