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Updated: Mar 26, 2026

Preparation and In Vivo Use of an Activity-based Probe for N-acylethanolamine Acid Amidase
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Potent α-amino-β-lactam carbamic acid ester as NAAA inhibitors. Synthesis and structure-activity relationship (SAR)

Andrea Nuzzi1, Annalisa Fiasella1, Jose Antonio Ortega1

  • 1Drug Discovery and Development, Italian Institute of Technology, Via Morego 30, I-16163 Genova, Italy.

European Journal of Medicinal Chemistry
|February 12, 2016
PubMed

Keywords:
CarbamatesCysteine hydrolaseInhibitorsN-acylethanolamine acid amidaseStructure–activity relationshipsβ-lactams

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