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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate

Craig W Lindsley, Kyle A Emmitte1, Corey R Hopkins

  • 1Department of Pharmaceutical Sciences, UNT System College of Pharmacy, University of North Texas Health Science Center , 3500 Camp Bowie Boulevard, Fort Worth, Texas 76107, United States.

Chemical Reviews
|February 17, 2016
PubMed

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