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SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists

Shuwen He1, Peter H Dobbelaar1, Liangqin Guo1

  • 1Early Development and Discovery Sciences, Merck Research Laboratories, 2000 Galloping Hill Road, Kenilworth, NJ 07033, United States.

Bioorganic & Medicinal Chemistry Letters
|February 23, 2016
PubMed

Keywords:
AntagonistSARSomatostatin receptor subtype 3Tetrahydro-β-carbolinehERG

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