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Structural optimization and structure-functional selectivity relationship studies of G protein-biased EP2 receptor

Seiji Ogawa1, Toshihide Watanabe1, Kazumi Moriyuki2

  • 1Medicinal Chemistry Research Laboratories, Ono Pharmaceutical Co., Ltd, 3-1-1 Sakurai, Shimamoto-cho, Mishima-gun, Osaka 618-8585, Japan.

Bioorganic & Medicinal Chemistry Letters
|April 9, 2016
PubMed

Keywords:
AgonistBiased ligandEP2ProstaglandinStructure–functional selectivity relationship

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