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Biosensor-based High Throughput Biopanning and Bioinformatics Analysis Strategy for the Global Validation of Drug-protein Interactions
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Target identification of covalently binding drugs by activity-based protein profiling (ABPP)

Christian M Pichler1, Joanna Krysiak2, Rolf Breinbauer1

  • 1Institute of Organic Chemistry, Graz University of Technology, Stremayrgasse 9, 8010 Graz, Austria.

Bioorganic & Medicinal Chemistry
|April 18, 2016
PubMed

Keywords:
Activity based protein profilingBiologically active moleculesCovalent binding drugsDrug targetsTarget identification

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