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Exploring new chemical functionalities to improve aromatase inhibition of steroids

Carla L Varela1, Cristina Amaral2, Georgina Correia-da-Silva2

  • 1Pharmaceutical Chemistry Group, Faculty of Pharmacy, University of Coimbra, 3000-548 Coimbra, Portugal.

Bioorganic & Medicinal Chemistry
|May 11, 2016
PubMed

Keywords:
Aromatase inhibitorsInduced-fit dockingMolecular modelingSteroidsStructure–activity relationshipsSynthesis

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