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Fragment-Based Discovery of 6-Arylindazole JAK Inhibitors

Andreas Ritzén1, Morten D Sørensen1, Kevin N Dack1

  • 1Drug Design, In Vitro Biology, Skin PK and Early Safety, and Preformulation & Early Analytical Development, Global R&D, LEO Pharma A/S , Industriparken 55, DK-2750 Ballerup, Denmark.

ACS Medicinal Chemistry Letters
|June 22, 2016
PubMed

Keywords:
FragmentsJAK inhibitorsindazolesphototoxicitypsoriasis

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