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Synthesis and evaluation of antitubercular activity of fluorinated 5-aryl-4-(hetero)aryl substituted pyrimidines

Egor V Verbitskiy1, Svetlana A Baskakova2, Marionella A Kravchenko3

  • 1Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, S. Kovalevskoy Str., 22, Ekaterinburg 620990, Russia; Ural Federal University, Mira St. 19, Ekaterinburg 620002, Russia.

Bioorganic & Medicinal Chemistry
|June 25, 2016
PubMed

Keywords:
AntimycobacterialCross-couplingNucleophilic aromatic substitution of hydrogenPyrimidineTuberculosis

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